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Accueil du site > Équipes > Résistance aux médicaments et protéines membranaires(P. Falson) > Publications

Publications

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2016 [Top] 10
280.  Atomic modelling and systematic mutagenesis identify residues in multiple drug binding sites that are essential for drug resistance in the major Candida transporter Cdr1.   
Nim S, Lobato LG, Moreno A, Chaptal V, Rawal MK, Falson P, Prasad R
(2016) Biochim Biophys Acta 1858 : 2858-2870

279.  Two different centered monoclinic crystals of the E. coli outer-membrane protein OmpF originate from the same building block.   
Chaptal V, Kilburg A, Flot D, Wiseman B, Aghajari N, Jault JM, Falson P
(2016) Biochim Biophys Acta 1858 : 326-32

278.  Overexpression, Membrane Preparation, and Purification of a Typical Multidrug ABC Transporter BmrA.   
Wiseman B, Jault JM
(2016) Methods Mol Biol 1432 : 133-42

277.  The linker region of breast cancer resistance protein ABCG2 is critical for coupling of ATP-dependent drug transport.   
Macalou S, Robey RW, Jabor Gozzi G, Shukla S, Grosjean I, Hegedus T, Ambudkar SV, Bates SE, Di Pietro A
(2016) Cell Mol Life Sci 73 : 1927-37

276.  Diffraction anisotropy falloff in the direction of the detergent belt for two centered monoclinic crystals of OmpF.   
Chaptal V, Kilburg A, Flot D, Wiseman B, Aghajari N, Jault JM, Falson P
(2016) Data Brief 7 : 726-9

275.  Single Nanoparticle Plasmonic Spectroscopy for Study of the Efflux Function of Multidrug ABC Membrane Transporters of Single Live Cells.   
Browning LM, Lee KJ, Cherukuri PK, Nallathamby PD, Warren S, Jault JM, Xu XN
(2016) RSC Adv 6 : 36794-36802

274.  2-Indolylmethylenebenzofuranones as first effective inhibitors of ABCC2.   
Baiceanu E, Nguyen KA, Gonzalez-Lobato L, Nasr R, Baubichon-Cortay H, Loghin F, Le Borgne M, Chow L, Boumendjel A, Peuchmaur M, Falson P
(2016) Eur J Med Chem 122 : 408-18

273.  pHluorin enables insights into the transport mechanism of antiporter Mdr1: R215 is critical for drug/H+ antiport.   
Redhu AK, Khandelwal NK, Banerjee A, Moreno A, Falson P, Prasad R
(2016) Biochem J 473 : 3127-45

272.  Leishmania tarentolae as a Promising Tool for Expressing Polytopic and Multi-Transmembrane Spans Eukaryotic Membrane Proteins: The Case of the ABC Pump ABCG6.   
Gonzalez-Lobato L, Chaptal V, Molle J, Falson P
(2016) Methods Mol Biol 1432 : 119-31

271.  Deciphering the molecular mechanisms underlying the binding of the TWIST1/E12 complex to regulatory E-box sequences.   
Bouard C, Terreux R, Honorat M, Manship B, Ansieau S, Vigneron AM, Puisieux A, Payen L
(2016) Nucleic Acids Res 44 : 5470-89

2015 [Top] 15
270.  Interaction between Bacillus subtilis YsxC and ribosomes (or rRNAs).   
Wicker-Planquart C, Jault JM
(2015) FEBS Lett 589 : 1026-32

269.  Autophosphorylation of the Bacterial Tyrosine-Kinase CpsD Connects Capsule Synthesis with the Cell Cycle in Streptococcus pneumoniae.   
Nourikyan J, Kjos M, Mercy C, Cluzel C, Morlot C, Noirot-Gros MF, Guiral S, Lavergne JP, Veening JW, Grangeasse C
(2015) PLoS Genet 11 : e1005518-e1005518

268.  Full engagement of liganded maltose-binding protein stabilizes a semi-open ATP-binding cassette dimer in the maltose transporter.   
Alvarez FJ, Orelle C, Huang Y, Bajaj R, Everly RM, Klug CS, Davidson AL
(2015) Mol Microbiol 98 : 878-94

267.  Downregulation of Toll-Like Receptor 9 Expression by Beta Human Papillomavirus 38 and Implications for Cell Cycle Control.   
Pacini L, Savini C, Ghittoni R, Saidj D, Lamartine J, Hasan UA, Accardi R, Tommasino M
(2015) J Virol 89 : 11396-405

266.  Protein synthesis by ribosomes with tethered subunits.   
Orelle C, Carlson ED, Szal T, Florin T, Jewett MC, Mankin AS
(2015) Nature 524 : 119-24

265.  Dual properties of hispidulin: antiproliferative effects on HepG2 cancer cells and selective inhibition of ABCG2 transport activity.   
Scoparo CT, Valdameri G, Worfel PR, Guterres FA, Martinez GR, Winnischofer SM, Di Pietro A, Rocha ME
(2015) Mol Cell Biochem 409 : 123-33

264.  A hydrophobic filter confers the cation selectivity of Zygosaccharomyces rouxii plasma-membrane Na+/H+ antiporter.   
Kinclova-Zimmermannova O, Falson P, Cmunt D, Sychrova H
(2015) J Mol Biol 427 : 1681-94

263.  Hepatitis C Virus Envelope Glycoprotein E1 Forms Trimers at the Surface of the Virion.   
Falson P, Bartosch B, Alsaleh K, Tews BA, Loquet A, Ciczora Y, Riva L, Montigny C, Montpellier C, Duverlie G, Pecheur EI, Le Maire M, Cosset FL, Dubuisson J, Penin F
(2015) J Virol 89 : 10333-46

262.  Recent trends of chalcones potentialities as antiproliferative and antiresistance agents.   
Winter E, Locatelli C, Di Pietro A, Creczynski-Pasa TB
(2015) Anticancer Agents Med Chem 15 : 592-604

261.  Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity.   
Gozzi GJ, Bouaziz Z, Winter E, Daflon-Yunes N, Honorat M, Guragossian N, Marminon C, Valdameri G, Bollacke A, Guillon J, Pinaud N, Marchivie M, Cadena SM, Jose J, Le Borgne M, Di Pietro A
(2015) Drug Des Devel Ther 9 : 3481-95

260.  The C-terminal ?-helix of YsxC is essential for its binding to 50S ribosome and rRNAs.   
Wicker-Planquart C, Ceres N, Jault JM
(2015) FEBS Lett 589 : 2080-6

259.  Quantification and kinetic study in plasma and tissues of (E)-1,1,4,4-tetramethyl-2-tetrazene, a liquid propellant and a transformation product of 1,1-dimethyl hydrazine.   
Payen L, Honorat M, Bouard C, Jacob G, Terreux R, Delalu H, Labarthe E, Guitton J
(2015) Anal Bioanal Chem 407 : 6721-9

258.  Biologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds.   
Bouaziz Z, Issa S, Gentili J, Gratz A, Bollacke A, Kassack M, Jose J, Herfindal L, Gausdal G, Dskeland SO, Mullie C, Sonnet P, Desgrouas C, Taudon N, Valdameri G, Di Pietro A, Baitiche M, Le Borgne M
(2015) J Enzyme Inhib Med Chem 30 : 180-8

257.  Modulators of the human ABCC2: hope from natural sources?   
Baiceanu E, Crisan G, Loghin F, Falson P
(2015) Future Med Chem 7 : 2041-63

256.  Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2.   
Jabor Gozzi G, Bouaziz Z, Winter E, Daflon-Yunes N, Aichele D, Nacereddine A, Marminon C, Valdameri G, Zeinyeh W, Bollacke A, Guillon J, Lacoudre A, Pinaud N, Cadena SM, Jose J, Le Borgne M, Di Pietro A
(2015) J Med Chem 58 : 265-77

2014 [Top] 13
255.  Identification of specific reversal agents for Leishmania ABCI4-mediated antimony resistance by flavonoid and trolox derivative screening.   
Manzano JI, Lecerf-Schmidt F, Lespinasse MA, Di Pietro A, Castanys S, Boumendjel A, Gamarro F
(2014) J Antimicrob Chemother 69 : 664-72

254.  Quinoxaline-substituted chalcones as new inhibitors of breast cancer resistance protein ABCG2: polyspecificity at B-ring position.   
Winter E, Gozzi GJ, Chiaradia-Delatorre LD, Daflon-Yunes N, Terreux R, Gauthier C, Mascarello A, Leal PC, Cadena SM, Yunes RA, Nunes RJ, Creczynski-Pasa TB, Di Pietro A
(2014) Drug Des Devel Ther 8 : 609-19

253.  Targeting the Achilles heel of multidrug-resistant cancer by exploiting the fitness cost of resistance.   
Szakacs G, Hall MD, Gottesman MM, Boumendjel A, Kachadourian R, Day BJ, Baubichon-Cortay H, Di Pietro A
(2014) Chem Rev 114 : 5753-74

252.  Understanding polyspecificity within the substrate-binding cavity of the human multidrug resistance P-glycoprotein.   
Martinez L, Arnaud O, Henin E, Tao H, Chaptal V, Doshi R, Andrieu T, Dussurgey S, Tod M, Di Pietro A, Zhang Q, Chang G, Falson P
(2014) FEBS J 281 : 673-82

251.  Mitochondrial metabolomics using high-resolution Fourier-transform mass spectrometry.   
Go YM, Uppal K, Walker DI, Tran V, Dury L, Strobel FH, Baubichon-Cortay H, Pennell KD, Roede JR, Jones DP
(2014) Methods Mol Biol 1198 : 43-73

250.  Quantitative evaluation of the combination between cytotoxic drug and efflux transporter inhibitors based on a tumour growth inhibition model.   
Sostelly A, Payen L, Guitton J, Di Pietro A, Falson P, Honorat M, Boumendjel A, Geze A, Freyer G, Tod M
(2014) Fundam Clin Pharmacol 28 : 161-9

249.  Jatrophanes from Euphorbia squamosa as potent inhibitors of Candida albicans multidrug transporters.   
Rawal MK, Shokoohinia Y, Chianese G, Zolfaghari B, Appendino G, Taglialatela-Scafati O, Prasad R, Di Pietro A
(2014) J Nat Prod 77 : 2700-6

248.  Collateral sensitivity of resistant MRP1-overexpressing cells to flavonoids and derivatives through GSH efflux.   
Lorendeau D, Dury L, Genoux-Bastide E, Lecerf-Schmidt F, Simoes-Pires C, Carrupt PA, Terreux R, Magnard S, Di Pietro A, Boumendjel A, Baubichon-Cortay H
(2014) Biochem Pharmacol 90 : 235-45

247.  Efficient and stable reconstitution of the ABC transporter BmrA for solid-state NMR studies.   
Kunert B, Gardiennet C, Lacabanne D, Calles-Garcia D, Falson P, Jault JM, Meier BH, Penin F, Bockmann A
(2014) Front Mol Biosci 1 : 5-5

246.  MBL-II-141, a chromone derivative, enhances irinotecan (CPT-11) anticancer efficiency in ABCG2-positive xenografts.   
Payen L, Honorat M, Guitton J, Gauthier C, Bouard C, Lecerf-Schmidt F, Peres B, Terreux R, Gervot H, Rioufol C, Boumendjel A, Puisieux A, Di Pietro A
(2014) Oncotarget 5 : 11957-70

245.  Symmetric bis-chalcones as a new type of breast cancer resistance protein inhibitors with a mechanism different from that of chromones.   
Winter E, Devantier Neuenfeldt P, Chiaradia-Delatorre LD, Gauthier C, Yunes RA, Nunes RJ, Creczynski-Pasa TB, Di Pietro A
(2014) J Med Chem 57 : 2930-41

244.  Stubborn contaminants: influence of detergents on the purity of the multidrug ABC transporter BmrA.   
Wiseman B, Kilburg A, Chaptal V, Reyes-Mejia GC, Sarwan J, Falson P, Jault JM
(2014) PLoS One 9 : e114864-e114864

243.  3D cryo-electron reconstruction of BmrA, a bacterial multidrug ABC transporter in an inward-facing conformation and in a lipidic environment.   
Fribourg PF, Chami M, Sorzano CO, Gubellini F, Marabini R, Marco S, Jault JM, Levy D
(2014) J Mol Biol 426 : 2059-69

2013 [Top] 16
242.  Sedimentation velocity analytical ultracentrifugation in hydrogenated and deuterated solvents for the characterization of membrane proteins.   
Le Roy A, Nury H, Wiseman B, Sarwan J, Jault JM, Ebel C
(2013) Methods Mol Biol 1033 : 219-51

241.  Regulatory interactions between a bacterial tyrosine kinase and its cognate phosphatase.   
Temel DB, Dutta K, Alphonse S, Nourikyan J, Grangeasse C, Ghose R
(2013) J Biol Chem 288 : 15212-28

240.  Structures of P-glycoprotein reveal its conformational flexibility and an epitope on the nucleotide-binding domain.   
Ward AB, Szewczyk P, Grimard V, Lee CW, Martinez L, Doshi R, Caya A, Villaluz M, Pardon E, Cregger C, Swartz DJ, Falson PG, Urbatsch IL, Govaerts C, Steyaert J, Chang G
(2013) Proc Natl Acad Sci U S A 110 : 13386-91

239.  A template model for studying anticancer drug efflux transporter inhibitors in vitro.   
Sostelly A, Payen L, Guitton J, Di Pietro A, Falson P, Honorat M, Valdameri G, Geze A, Boumendjel A, Freyer G, Tod M
(2013) Fundam Clin Pharmacol 27 : 544-56

238.  Comparative analysis of the Tyr-kinases CapB1 and CapB2 fused to their cognate modulators CapA1 and CapA2 from Staphylococcus aureus.   
Gruszczyk J, Olivares-Illana V, Nourikyan J, Fleurie A, Bechet E, Gueguen-Chaignon V, Freton C, Aumont-Nicaise M, Morera S, Grangeasse C, Nessler S
(2013) PLoS One 8 : e75958-e75958

237.  ABCG2 is not able to catalyze glutathione efflux and does not contribute to GSH-dependent collateral sensitivity.   
Gauthier C, Ozvegy-Laczka C, Szakacs G, Sarkadi B, Di Pietro A
(2013) Front Pharmacol 4 : 138-138

236.  New structure-activity relationships of chalcone inhibitors of breast cancer resistance protein: polyspecificity toward inhibition and critical substitutions against cytotoxicity.   
Rangel LP, Winter E, Gauthier C, Terreux R, Chiaradia-Delatorre LD, Mascarello A, Nunes RJ, Yunes RA, Creczynski-Pasa TB, Macalou S, Lorendeau D, Baubichon-Cortay H, Ferreira-Pereira A, Di Pietro A
(2013) Drug Des Devel Ther 7 : 1043-52

235.  ABCG2: recent discovery of potent and highly selective inhibitors.   
Lecerf-Schmidt F, Peres B, Valdameri G, Gauthier C, Winter E, Payen L, Di Pietro A, Boumendjel A
(2013) Future Med Chem 5 : 1037-45

234.  Modular construction of quaternary hemiaminal-based inhibitor candidates and their in cellulo assessment with HIV-1 protease.   
Gros G, Martinez L, Gimenez AS, Adler P, Maurin P, Wolkowicz R, Falson P, Hasserodt J
(2013) Bioorg Med Chem 21 : 5407-13

233.  Structure-activity relationships of chromone derivatives toward the mechanism of interaction with and inhibition of breast cancer resistance protein ABCG2.   
Winter E, Lecerf-Schmidt F, Gozzi G, Peres B, Lightbody M, Gauthier C, Ozvegy-Laczka C, Szakacs G, Sarkadi B, Creczynski-Pasa TB, Boumendjel A, Di Pietro A
(2013) J Med Chem 56 : 9849-60

232.  Tools for characterizing bacterial protein synthesis inhibitors.   
Orelle C, Carlson S, Kaushal B, Almutairi MM, Liu H, Ochabowicz A, Quan S, Pham VC, Squires CL, Murphy BT, Mankin AS
(2013) Antimicrob Agents Chemother 57 : 5994-6004

231.  Azaindole derivatives are inhibitors of microtubule dynamics, with anti-cancer and anti-angiogenic activities.   
Prudent R, Vassal-Stermann E, Nguyen CH, Mollaret M, Viallet J, Desroches-Castan A, Martinez A, Barette C, Pillet C, Valdameri G, Soleilhac E, Di Pietro A, Feige JJ, Billaud M, Florent JC, Lafanechere L
(2013) Br J Pharmacol 168 : 673-85

230.  Small angle neutron scattering for the study of solubilised membrane proteins.   
Breyton C, Gabel F, Lethier M, Flayhan A, Durand G, Jault JM, Juillan-Binard C, Imbert L, Moulin M, Ravaud S, Hartlein M, Ebel C
(2013) Eur Phys J E Soft Matter 36 : 71-71

229.  Localization of putative binding sites for cyclic guanosine monophosphate and the anti-cancer drug 5-fluoro-2'-deoxyuridine-5'-monophosphate on ABCC11 in silico models.   
Honorat M, Terreux R, Falson P, Di Pietro A, Dumontet C, Payen L
(2013) BMC Struct Biol 13 : 7-7

228.  Characterization of hydrophobic peptides in the presence of detergent by photoionization mass spectrometry.   
Bagag A, Jault JM, Sidahmed-Adrar N, Refregiers M, Giuliani A, Le Naour F
(2013) PLoS One 8 : e79033-e79033

227.  Identifying the targets of aminoacyl-tRNA synthetase inhibitors by primer extension inhibition.   
Orelle C, Szal T, Klepacki D, Shaw KJ, Vazquez-Laslop N, Mankin AS
(2013) Nucleic Acids Res 41 : e144-e144

2012 [Top] 15
226.  PatA and PatB form a functional heterodimeric ABC multidrug efflux transporter responsible for the resistance of Streptococcus pneumoniae to fluoroquinolones.   
Boncoeur E, Durmort C, Bernay B, Ebel C, Di Guilmi AM, Croize J, Vernet T, Jault JM
(2012) Biochemistry 51 : 7755-65

225.  Potassium acts as a GTPase-activating element on each nucleotide-binding domain of the essential Bacillus subtilis EngA.   
Foucher AE, Reiser JB, Ebel C, Housset D, Jault JM
(2012) PLoS One 7 : e46795-e46795

224.  Substituted chromones as highly potent nontoxic inhibitors, specific for the breast cancer resistance protein.   
Valdameri G, Genoux-Bastide E, Peres B, Gauthier C, Guitton J, Terreux R, Winnischofer SM, Rocha ME, Boumendjel A, Di Pietro A
(2012) J Med Chem 55 : 966-70

223.  Methoxy stilbenes as potent, specific, untransported, and noncytotoxic inhibitors of breast cancer resistance protein.   
Valdameri G, Pereira Rangel L, Spatafora C, Guitton J, Gauthier C, Arnaud O, Ferreira-Pereira A, Falson P, Winnischofer SM, Rocha ME, Tringali C, Di Pietro A
(2012) ACS Chem Biol 7 : 322-30

222.  A synthetic chalcone as a potent inducer of glutathione biosynthesis.   
Kachadourian R, Day BJ, Pugazhenti S, Franklin CC, Genoux-Bastide E, Mahaffey G, Gauthier C, Di Pietro A, Boumendjel A
(2012) J Med Chem 55 : 1382-8

221.  Bridging the gap between structure and kinetics of human SGLT1.   
Sala-Rabanal M, Hirayama BA, Loo DD, Chaptal V, Abramson J, Wright EM
(2012) Am J Physiol Cell Physiol 302 : C1293-305

220.  Phosphorylation of CpgA protein enhances both its GTPase activity and its affinity for ribosome and is crucial for Bacillus subtilis growth and morphology.   
Pompeo F, Freton C, Wicker-Planquart C, Grangeasse C, Jault JM, Galinier A
(2012) J Biol Chem 287 : 20830-8

219.  Stoichiometry of the MexA-OprM binding, as investigated by blue native gel electrophoresis.   
Ferrandez Y, Monlezun L, Phan G, Benabdelhak H, Benas P, Ulryck N, Falson P, Ducruix A, Picard M, Broutin I
(2012) Electrophoresis 33 : 1282-7

218.  Investigation of chalcones as selective inhibitors of the breast cancer resistance protein: critical role of methoxylation in both inhibition potency and cytotoxicity.   
Valdameri G, Gauthier C, Terreux R, Kachadourian R, Day BJ, Winnischofer SM, Rocha ME, Frachet V, Ronot X, Di Pietro A, Boumendjel A
(2012) J Med Chem 55 : 3193-200

217.  Ex vivo and in vivo inhibition of human rhinovirus replication by a new pseudosubstrate of viral 2A protease.   
Falah N, Violot S, Decimo D, Berri F, Foucault-Grunenwald ML, Ohlmann T, Schuffenecker I, Morfin F, Lina B, Riteau B, Cortay JC
(2012) J Virol 86 : 691-704

216.  Pharmacological inhibition of LIM kinase stabilizes microtubules and inhibits neoplastic growth.   
Prudent R, Vassal-Stermann E, Nguyen CH, Pillet C, Martinez A, Prunier C, Barette C, Soleilhac E, Filhol O, Beghin A, Valdameri G, Honore S, Aci-Seche S, Grierson D, Antonipillai J, Li R, Di Pietro A, Dumontet C, Braguer D, Florent JC, Knapp S, Bernard O, Lafanechere L
(2012) Cancer Res 72 : 4429-39

215.  Microparticle-mediated transfer of the viral receptors CAR and CD46, and the CFTR channel in a CHO cell model confers new functions to target cells.   
Gonzalez G, Vituret C, Di Pietro A, Chanson M, Boulanger P, Hong SS
(2012) PLoS One 7 : e52326-e52326

214.  Blocking human enterovirus 71 replication by targeting viral 2A protease.   
Falah N, Montserret R, Lelogeais V, Schuffenecker I, Lina B, Cortay JC, Violot S
(2012) J Antimicrob Chemother 67 : 2865-9

213.  Dynamics of a bacterial multidrug ABC transporter in the inward- and outward-facing conformations.   
Mehmood S, Domene C, Forest E, Jault JM
(2012) Proc Natl Acad Sci U S A 109 : 10832-6

212.  6-halogenochromones bearing tryptamine: one-step access to potent and highly selective inhibitors of breast cancer resistance protein.   
Valdameri G, Genoux-Bastide E, Gauthier C, Peres B, Terreux R, Winnischofer SM, Rocha ME, Di Pietro A, Boumendjel A
(2012) ChemMedChem 7 : 1177-80

2011 [Top] 12
211.  MRP8/ABCC11 expression is regulated by dexamethasone in breast cancer cells and is associated to progesterone receptor status in breast tumors.   
Honorat M, Mesnier A, Vendrell J, Di Pietro A, Lin V, Dumontet C, Cohen P, Payen L
(2011) Int J Breast Cancer 2011 : 807380-807380

210.  Crystal structure of lactose permease in complex with an affinity inactivator yields unique insight into sugar recognition.     
Chaptal V, Kwon S, Sawaya MR, Guan L, Kaback HR, Abramson J
(2011) Proc Natl Acad Sci U S A 108 : 9361-6

209.  Identification of xanthones as selective killers of cancer cells overexpressing the ABC transporter MRP1.   
Genoux-Bastide E, Lorendeau D, Nicolle E, Yahiaoui S, Magnard S, Di Pietro A, Baubichon-Cortay H, Boumendjel A
(2011) ChemMedChem 6 : 1478-84

208.  Dicer-mediated upregulation of BCRP confers tamoxifen resistance in human breast cancer cells.   
Selever J, Gu G, Lewis MT, Beyer A, Herynk MH, Covington KR, Tsimelzon A, Dontu G, Provost P, Di Pietro A, Boumendjel A, Albain K, Miele L, Weiss H, Barone I, Ando S, Fuqua SA
(2011) Clin Cancer Res 17 : 6510-21

207.  Binding, reconstitution and 2D crystallization of membrane or soluble proteins onto functionalized lipid layer observed in situ by reflected light microscopy.   
Dezi M, Fribourg PF, Cicco AD, Jault JM, Chami M, Levy D
(2011) J Struct Biol 174 : 307-14

206.  Optimized purification of a heterodimeric ABC transporter in a highly stable form amenable to 2-D crystallization.   
Galian C, Manon F, Dezi M, Torres C, Ebel C, Levy D, Jault JM
(2011) PLoS One 6 : e19677-e19677

205.  Targeting the multidrug ABCG2 transporter with flavonoidic inhibitors: in vitro optimization and in vivo validation.   
Boumendjel A, Macalou S, Valdameri G, Pozza A, Gauthier C, Arnaud O, Nicolle E, Magnard S, Falson P, Terreux R, Carrupt PA, Payen L, Di Pietro A
(2011) Curr Med Chem 18 : 3387-401

204.  Structuring detergents for extracting and stabilizing functional membrane proteins.     
Matar-Merheb R, Rhimi M, Leydier A, Huche F, Galian C, Desuzinges-Mandon E, Ficheux D, Flot D, Aghajari N, Kahn R, Di Pietro A, Jault JM, Coleman AW, Falson P
(2011) PLoS One 6 : e18036-e18036

203.  The acridone derivative MBLI-87 sensitizes breast cancer resistance protein-expressing xenografts to irinotecan.     
Arnaud O, Boumendjel A, Geze A, Honorat M, Matera EL, Guitton J, Stein WD, Bates SE, Falson P, Dumontet C, Di Pietro A, Payen L
(2011) Eur J Cancer 47 : 640-8

202.  Leucine-rich protein 130 contributes to apoptosis resistance of human hepatocarcinoma cells.     
Michaud M, Barakat S, Magnard S, Rigal D, Baggetto LG
(2011) Int J Oncol 38 : 169-78

201.  Crenarchaeal CdvA forms double-helical filaments containing DNA and interacts with ESCRT-III-like CdvB.   
Moriscot C, Gribaldo S, Jault JM, Krupovic M, Arnaud J, Jamin M, Schoehn G, Forterre P, Weissenhorn W, Renesto P
(2011) PLoS One 6 : e21921-e21921

200.  Multidrug resistance ABC transporter structure predictions by homology modeling approaches.     
Honorat M, Falson P, Terreux R, Di Pietro A, Dumontet C, Payen L
(2011) Curr Drug Metab 12 : 268-77

2010 [Top] 16
199.  The mechanism of sodium and substrate release from the binding pocket of vSGLT.     
Watanabe A, Choe S, Chaptal V, Rosenberg JM, Wright EM, Grabe M, Abramson J
(2010) Nature 468 : 988-91

198.  Magnesium dependent complexation of tri-anionic calix[4]arene detergents by the nucleotide binding domain 1 (NBD1) of multidrug resistance protein MRP1     
Nault LFA, Girardot C, Leydier A, Coleman AW, Perrotton T, Magnard S, Baubichon-Cortay H
(2010) NEW JOURNAL OF CHEMISTRY 34 : 1812-1815

197.  Potent and fully noncompetitive peptidomimetic inhibitor of multidrug resistance P-glycoprotein.     
Arnaud O, Koubeissi A, Ettouati L, Terreux R, Alame G, Grenot C, Dumontet C, Di Pietro A, Paris J, Falson P
(2010) J Med Chem 53 : 6720-9

196.  Dynamics of alpha-helical subdomain rotation in the intact maltose ATP-binding cassette transporter.   
Orelle C, Alvarez FJ, Oldham ML, Orelle A, Wiley TE, Chen J, Davidson AL
(2010) Proc Natl Acad Sci U S A 107 : 20293-8

195.  Hijacking of the pleiotropic cytokine interferon-? by the type III secretion system of Yersinia pestis.   
Gendrin C, Sarrazin S, Bonnaffe D, Jault JM, Lortat-Jacob H, Dessen A
(2010) PLoS One 5 : e15242-e15242

194.  Rapid readout detector captures protein time-resolved WAXS.     
Westenhoff S, Malmerberg E, Arnlund D, Johansson L, Nazarenko E, Cammarata M, Davidsson J, Chaptal V, Abramson J, Katona G, Menzel A, Neutze R
(2010) Nat Methods 7 : 775-6

193.  Iodination of verapamil for a stronger induction of death, through GSH efflux, of cancer cells overexpressing MRP1.     
Barattin R, Perrotton T, Trompier D, Lorendeau D, Di Pietro A, D'Hardemare Adu M, Baubichon-Cortay H
(2010) Bioorg Med Chem 18 : 6265-74

192.  Insect cell versus bacterial overexpressed membrane proteins: an example, the human ABCG2 transporter.   
Pozza A, Perez-Victoria JM, Di Pietro A
(2010) Methods Mol Biol 654 : 47-75

191.  Multiple effects of silymarin on the hepatitis C virus lifecycle.     
Wagoner J, Negash A, Kane OJ, Martinez LE, Nahmias Y, Bourne N, Owen DM, Grove J, Brimacombe C, McKeating JA, Pecheur EI, Graf TN, Oberlies NH, Lohmann V, Cao F, Tavis JE, Polyak SJ
(2010) Hepatology 51 : 1912-21

190.  The multidrug resistance half-transporter ABCG2 is purified as a tetramer upon selective extraction from membranes.     
Dezi M, Fribourg PF, Di Cicco A, Arnaud O, Marco S, Falson P, Di Pietro A, Levy D
(2010) Biochim Biophys Acta 1798 : 2094-101

189.  Functional reconstitution of an ABC transporter in nanodiscs for use in electron paramagnetic resonance spectroscopy.   
Alvarez FJ, Orelle C, Davidson AL
(2010) J Am Chem Soc 132 : 9513-5

188.  Gated access to the pore of a P2X receptor: structural implications for closed-open transitions.     
Kracun S, Chaptal V, Abramson J, Khakh BS
(2010) J Biol Chem 285 : 10110-21

187.  Mammalian membrane protein expression in baculovirus-infected insect cells.   
Trometer C, Falson P
(2010) Methods Mol Biol 601 : 105-17

186.  ABCG2 transports and transfers heme to albumin through its large extracellular loop.     
Desuzinges-Mandon E, Arnaud O, Martinez L, Huche F, Di Pietro A, Falson P
(2010) J Biol Chem 285 : 33123-33

185.  Fluorescence Detection of Heavy Atom Labeling (FD-HAL): A rapid method for identifying covalently modified cysteine residues by phasing atoms     
Chaptal V, Ujwal R, Nie YL, Watanabe A, Kwon S, Abramson J
(2010) JOURNAL OF STRUCTURAL BIOLOGY 171 : 82-87

184.  Fluorescence Detection of Heavy Atom Labeling (FD-HAL): a rapid method for identifying covalently modified cysteine residues by phasing atoms.   
Chaptal V, Ujwal R, Nie Y, Watanabe A, Kwon S, Abramson J
(2010) J Struct Biol 171 : 82-7

2009 [Top] 15
183.  The ATPase activity of an 'essential' Bacillus subtilis enzyme, YdiB, is required for its cellular function and is modulated by oligomerization.   
Karst JC, Foucher AE, Campbell TL, Di Guilmi AM, Stroebel D, Mangat CS, Brown ED, Jault JM
(2009) Microbiology 155 : 944-56

182.  The YheI/YheH heterodimer from Bacillus subtilis is a multidrug ABC transporter.   
Torres C, Galian C, Freiberg C, Fantino JR, Jault JM
(2009) Biochim Biophys Acta 1788 : 615-22

181.  Crystal packing analysis of murine VDAC1 crystals in a lipidic environment reveals novel insights on oligomerization and orientation.   
Ujwal R, Cascio D, Chaptal V, Ping P, Abramson J
(2009) Channels (Austin) 3 : 167-70

180.  Overexpression of homogeneous and active ABCG2 in insect cells.     
Pozza A, Perez-Victoria JM, Prez-Victoria JM, Di Pietro A
(2009) Protein Expr Purif 63 : 75-83

179.  Becatecarin (rebeccamycin analog, NSC 655649) is a transport substrate and induces expression of the ATP-binding cassette transporter, ABCG2, in lung carcinoma cells.     
Robey RW, Obrzut T, Shukla S, Polgar O, Macalou S, Bahr JC, Di Pietro A, Ambudkar SV, Bates SE
(2009) Cancer Chemother Pharmacol 64 : 575-83

178.  A 3D linear solvation energy model to quantify the affinity of flavonoid derivatives toward P-glycoprotein.     
Boccard J, Bajot F, Di Pietro A, Rudaz S, Boumendjel A, Nicolle E, Carrupt PA
(2009) Eur J Pharm Sci 36 : 254-64

177.  Structure and functional analysis of a Ca2+ sensor mutant of the Na+/Ca2+ exchanger.     
Chaptal V, Ottolia M, Mercado-Besserer G, Nicoll DA, Philipson KD, Abramson J
(2009) J Biol Chem 284 : 14688-92

176.  Keeping an eye on membrane transport by TR-WAXS.     
Abramson J, Chaptal V
(2009) Structure 17 : 1153-5

175.  Breast cancer resistance protein (BCRP/ABCG2): new inhibitors and QSAR studies by a 3D linear solvation energy approach.     
Nicolle E, Boccard J, Guilet D, Dijoux-Franca MG, Zelefac F, Macalou S, Grosselin J, Schmidt J, Carrupt PA, Di Pietro A, Boumendjel A
(2009) Eur J Pharm Sci 38 : 39-46

174.  The ATPase activity of an 'essential' Bacillus subtilis enzyme, YdiB, is required for its cellular function and is modulated by oligomerization   
Karst JC, Foucher AE, Campbell TL, Di Guilmi AM, Stroebel D,Managat CS,Brown ED, Jault JM
(2009) MICROBIOLOGY-SGM 155 : 944-956

173.  Alternating access in maltose transporter mediated by rigid-body rotations.   
Khare D, Oldham ML, Orelle C, Davidson AL, Chen J
(2009) Mol Cell 33 : 528-36

172.  QSAR analysis and molecular modeling of ABCG2-specific inhibitors.     
Nicolle E, Boumendjel A, Macalou S, Genoux E, Ahmed-Belkacem A, Carrupt PA, Di Pietro A
(2009) Adv Drug Deliv Rev 61 : 34-46

171.  Probing the conformation of the resting state of a bacterial multidrug ABC transporter, BmrA, by a site-directed spin labeling approach.     
Do Cao MA, Crouzy S, Kim M, Becchi M, Cafiso DS, Di Pietro A, Jault JM
(2009) Protein Sci 18 : 1507-20

170.  Jatrophane diterpenes from Euphorbia spp. as modulators of multidrug resistance in cancer therapy     
Corea G, Di Pietro A, Dumontet C, Fattorusso E, Lanzotti V
(2009) PHYTOCHEMISTRY REVIEWS 8 : 431-447

169.  Selective modulation of P-glycoprotein activity by steroidal saponines from Paris polyphylla.     
Nguyen VT, Darbour N, Bayet C, Doreau A, Raad I, Phung BH, Dumontet C, Di Pietro A, Dijoux-Franca MG, Guilet D
(2009) Fitoterapia 80 : 39-42

2008 [Top] 9
168.  Crystal structure and functional analysis identify the P-loop containing protein YFH7 of Saccharomyces cerevisiae as an ATP-dependent kinase.     
Gueguen-Chaignon V, Chaptal V, Lariviere L, Costa N, Lopes P, Morera S, Nessler S
(2008) Proteins 71 : 804-12

167.  Structure, function, and evolution of bacterial ATP-binding cassette systems.   
Davidson AL, Dassa E, Orelle C, Chen J
(2008) Microbiol Mol Biol Rev 72 : 317contents-364contents

166.  ABCC11 expression is regulated by estrogen in MCF7 cells, correlated with estrogen receptor alpha expression in postmenopausal breast tumors and overexpressed in tamoxifen-resistant breast cancer cells.   
Honorat M, Mesnier A, Vendrell J, Guitton J, Bieche I, Lidereau R, Kruh GD, Dumontet C, Cohen P, Payen L
(2008) Endocr Relat Cancer 15 : 125-38

165.  Discovery of a new series of jatrophane and lathyrane diterpenes as potent and specific P-glycoprotein modulators.     
Barile E, Borriello M, Di Pietro A, Doreau A, Fattorusso C, Fattorusso E, Lanzotti V
(2008) Org Biomol Chem 6 : 1756-62

164.  Both maltose-binding protein and ATP are required for nucleotide-binding domain closure in the intact maltose ABC transporter.   
Orelle C, Ayvaz T, Everly RM, Klug CS, Davidson AL
(2008) Proc Natl Acad Sci U S A 105 : 12837-42

163.  Conformational change induced by ATP binding in the multidrug ATP-binding cassette transporter BmrA.     
Orelle C, Gubellini F, Durand A, Marco S, Levy D, Gros P, Di Pietro A, Jault JM
(2008) Biochemistry 47 : 2404-12

162.  Dexamethasone down-regulates ABCG2 expression levels in breast cancer cells.     
Honorat M, Mesnier A, Di Pietro A, Lin V, Cohen P, Dumontet C, Payen L
(2008) Biochem Biophys Res Commun 375 : 308-14

161.  Trianionic calix[4]arene monoalkoxy derivatives: synthesis, solid-state structures and self-assembly properties     
Suwinska K, Shkurenko O, Mbemba C, Leydier A, Jebors S, Coleman AW, Matar R, Falson P
(2008) NEW JOURNAL OF CHEMISTRY 32 : 1988-1998

160.  Interactions of an essential Bacillus subtilis GTPase, YsxC, with ribosomes.   
Wicker-Planquart C, Foucher AE, Louwagie M, Britton RA, Jault JM
(2008) J Bacteriol 190 : 681-90

2007 [Top] 8
159.  Acridone derivatives: design, synthesis, and inhibition of breast cancer resistance protein ABCG2.     
Boumendjel A, Macalou S, Ahmed-Belkacem A, Blanc M, Di Pietro A
(2007) Bioorg Med Chem 15 : 2892-7

158.  Structural analysis of the bacterial HPr kinase/phosphorylase V267F mutant gives insights into the allosteric regulation mechanism of this bifunctional enzyme.     
Chaptal V, Vincent F, Gueguen-Chaignon V, Monedero V, Poncet S, Deutscher J, Nessler S, Morera S
(2007) J Biol Chem 282 : 34952-7

157.  How does regulatory Ca2+ regulate the Na+-Ca2+ exchanger?   
Chaptal V, Besserer GM, Ottolia M, Nicoll DA, Cascio D, Philipson KD, Abramson J
(2007) Channels (Austin) 1 : 397-9

156.  Influence of tyrosine-kinase Wzc activity on colanic acid production in Escherichia coli K12 cells.     
Obadia B, Lacour S, Doublet P, Baubichon-Cortay H, Cozzone AJ, Grangeasse C
(2007) J Mol Biol 367 : 42-53

155.  Tyrosine-kinase Wzc from Escherichia coli possesses an ATPase activity regulated by autophosphorylation.     
Soulat D, Jault JM, Geourjon C, Gouet P, Cozzone AJ, Grangeasse C
(2007) FEMS Microbiol Lett 274 : 252-9

154.  Nonprenylated rotenoids, a new class of potent breast cancer resistance protein inhibitors.     
Ahmed-Belkacem A, Macalou S, Borrelli F, Capasso R, Fattorusso E, Taglialatela-Scafati O, Di Pietro A
(2007) J Med Chem 50 : 1933-8

153.  (R)- and (S)-verapamil differentially modulate the multidrug-resistant protein MRP1.     
Perrotton T, Trompier D, Chang XB, Di Pietro A, Baubichon-Cortay H
(2007) J Biol Chem 282 : 31542-8

152.  The second Ca2+-binding domain of the Na+ Ca2+ exchanger is essential for regulation: crystal structures and mutational analysis.     
Besserer GM, Ottolia M, Nicoll DA, Chaptal V, Cascio D, Philipson KD, Abramson J
(2007) Proc Natl Acad Sci U S A 104 : 18467-72

2006 [Top] 10
151.  Multiple GTPases participate in the assembly of the large ribosomal subunit in Bacillus subtilis.   
Schaefer L, Uicker WC, Wicker-Planquart C, Foucher AE, Jault JM, Britton RA
(2006) J Bacteriol 188 : 8252-8

150.  Structural analysis of B. subtilis CcpA effector binding site.     
Chaptal V, Gueguen-Chaignon V, Poncet S, Lecampion C, Meyer P, Deutscher J, Galinier A, Nessler S, Morera S
(2006) Proteins 64 : 814-6

149.  Conformational changes in sarcoplasmic reticulum Ca(2+)-ATPase mutants: effect of mutations either at Ca(2+)-binding site II or at tryptophan 552 in the cytosolic domain.     
Lenoir G, Jaxel C, Picard M, Le Maire M, Champeil P, Falson P
(2006) Biochemistry 45 : 5261-70

148.  Staphylococcus aureus operates protein-tyrosine phosphorylation through a specific mechanism.     
Soulat D, Jault JM, Duclos B, Geourjon C, Cozzone AJ, Grangeasse C
(2006) J Biol Chem 281 : 14048-56

147.  Purification of breast cancer resistance protein ABCG2 and role of arginine-482      
Pozza A, Perez-Victoria JM, Sardo A, Ahmed-Belkacem A, Di Pietro A
(2006) CELLULAR AND MOLECULAR LIFE SCIENCES  63 : 1912-1922

146.  Combination of suboptimal doses of inhibitors targeting different domains of LtrMDR1 efficiently overcomes resistance of Leishmania spp. to Miltefosine by inhibiting drug efflux.     
Perez-Victoria JM, Cortes-Selva F, Parodi-Talice A, Bavchvarov BI, Perez-Victoria FJ, Munoz-Martinez F, Maitrejean M, Costi MP, Barron D, Di Pietro A, Castanys S, Gamarro F
(2006) Antimicrob Agents Chemother 50 : 3102-10

145.  The ABC transporter BmrA from Bacillus subtilis is a functional dimer when in a detergent-solubilized state.     
Ravaud S, Do Cao MA, Jidenko M, Ebel C, Le Maire M, Jault JM, Di Pietro A, Haser R, Aghajari N
(2006) Biochem J 395 : 345-53

144.  X-ray structure of a domain-swapped dimer of Ser46-phosphorylated Crh from Bacillus subtilis.     
Chaptal V, Lariviere L, Gueguen-Chaignon V, Galinier A, Nessler S, Morera S
(2006) Proteins 63 : 249-51

143.  Inhibitors of cancer cell multidrug resistance mediated by breast cancer resistance protein (BCRP/ABCG2).     
Ahmed-Belkacem A, Pozza A, Macalou S, Perez-Victoria JM, Boumendjel A, Di Pietro A
(2006) Anticancer Drugs 17 : 239-43

142.  Role of the yeast ABC transporter Yor1p in cadmium detoxification.     
Nagy Z, Montigny C, Leverrier P, Yeh S, Goffeau A, Garrigos M, Falson P
(2006) Biochimie 88 : 1665-71

2005 [Top] 5
141.  Time-resolved fluorescence resonance energy transfer shows that the bacterial multidrug ABC half-transporter BmrA functions as a homodimer.     
Dalmas O, Do Cao MA, Lugo MR, Sharom FJ, Di Pietro A, Jault JM
(2005) Biochemistry 44 : 4312-21

140.  Anticancer multidrug resistance mediated by MRP1: recent advances in the discovery of reversal agents.     
Boumendjel A, Baubichon-Cortay H, Trompier D, Perrotton T, Di Pietro A
(2005) Med Res Rev 25 : 453-72

139.  Flavonoid structure-activity studies identify 6-prenylchrysin and tectochrysin as potent and specific inhibitors of breast cancer resistance protein ABCG2.     
Ahmed-Belkacem A, Pozza A, Munoz-Martinez F, Bates SE, Castanys S, Gamarro F, Di Pietro A, Perez-Victoria JM
(2005) Cancer Res 65 : 4852-60

138.  The binding mechanism of the yeast F1-ATPase inhibitory peptide: role of catalytic intermediates and enzyme turnover.     
Corvest V, Sigalat C, Venard R, Falson P, Mueller DM, Haraux F
(2005) J Biol Chem 280 : 9927-36

137.  The Q-loop disengages from the first intracellular loop during the catalytic cycle of the multidrug ABC transporter BmrA.     
Dalmas O, Orelle C, Foucher AE, Geourjon C, Crouzy S, Di Pietro A, Jault JM
(2005) J Biol Chem 280 : 36857-64

2004 [Top] 11
136.  A new method for the reconstitution of membrane proteins into giant unilamellar vesicles.     
Girard P, Pecreaux J, Lenoir G, Falson P, Rigaud JL, Bassereau P
(2004) Biophys J 87 : 419-29

135.  Jatrophane diterpenes as modulators of multidrug resistance. Advances of structure-activity relationships and discovery of the potent lead pepluanin A.     
Corea G, Fattorusso E, Lanzotti V, Motti R, Simon PN, Dumontet C, Di Pietro A
(2004) J Med Chem 47 : 988-92

134.  Involvement of the L6-7 loop in SERCA1a Ca2+-ATPase activation by Ca2+ (or Sr2+) and ATP.     
Lenoir G, Picard M, Mller JV, Le Maire M, Champeil P, Falson P
(2004) J Biol Chem 279 : 32125-33

133.  Characterization of YvcC (BmrA), a multidrug ABC transporter constitutively expressed in Bacillus subtilis.     
Steinfels E, Orelle C, Fantino JR, Dalmas O, Rigaud JL, Denizot F, Di Pietro A, Jault JM
(2004) Biochemistry 43 : 7491-502

132.  Two FHA domains on an ABC transporter, Rv1747, mediate its phosphorylation by PknF, a Ser/Thr protein kinase from Mycobacterium tuberculosis.     
Molle V, Soulat D, Jault JM, Grangeasse C, Cozzone AJ, Prost JF
(2004) FEMS Microbiol Lett 234 : 215-23

131.  HPr kinase/phosphorylase, a Walker motif A-containing bifunctional sensor enzyme controlling catabolite repression in Gram-positive bacteria.     
Poncet S, Mijakovic I, Nessler S, Gueguen-Chaignon V, Chaptal V, Galinier A, Boel G, Maze A, Deutscher J
(2004) Biochim Biophys Acta 1697 : 123-35

130.  Functional properties of sarcoplasmic reticulum Ca(2+)-ATPase after proteolytic cleavage at Leu119-Lys120, close to the A-domain.     
Lenoir G, Picard M, Gauron C, Montigny C, Le Marechal P, Falson P, Le Maire M, Mller JV, Champeil P
(2004) J Biol Chem 279 : 9156-66

129.  Structural insight into the cooperativity between catalytic and noncatalytic sites of F1-ATPase.     
Falson P, Goffeau A, Boutry M, Jault JM
(2004) Biochim Biophys Acta 1658 : 133-40

128.  Structure-activity relationships for euphocharacins A-L, a new series of jatrophane diterpenes, as inhibitors of cancer cell P-glycoprotein.     
Corea G, Fattorusso E, Lanzotti V, Motti R, Simon PN, Dumontet C, Di Pietro A
(2004) Planta Med 70 : 657-65

127.  Verapamil and its derivative trigger apoptosis through glutathione extrusion by multidrug resistance protein MRP1.     
Trompier D, Chang XB, Barattin R, Du Moulinet D'Hardemare A, Di Pietro A, Baubichon-Cortay H
(2004) Cancer Res 64 : 4950-6

126.  Overcoming the toxicity of membrane peptide expression in bacteria by upstream insertion of Asp-Pro sequence.     
Montigny C, Penin F, Lethias C, Falson P
(2004) Biochim Biophys Acta 1660 : 53-65

2003 [Top] 11
125.  Jatrophane diterpenes as P-glycoprotein inhibitors. First insights of structure-activity relationships and discovery of a new, powerful lead.     
Corea G, Fattorusso E, Lanzotti V, Taglialatela-Scafati O, Appendino G, Ballero M, Simon PN, Dumontet C, Di Pietro A
(2003) J Med Chem 46 : 3395-402

124.  Multiple flavonoid-binding sites within multidrug resistance protein MRP1.     
Trompier D, Baubichon-Cortay H, Chang XB, Maitrejean M, Barron D, Riordon JR, Di Pietro A
(2003) Cell Mol Life Sci 60 : 2164-77

123.  Potent competitive inhibition of drug binding to the Saccharomyces cerevisiae ABC exporter Pdr5p by the hydrophobic estradiol-derivative RU49953.     
Conseil G, Perez-Victoria JM, Renoir JM, Goffeau A, Di Pietro A
(2003) Biochim Biophys Acta 1614 : 131-4

122.  Involvement of the cytoplasmic loop L6-7 in the entry mechanism for transport of Ca2+ through the sarcoplasmic reticulum Ca2+-ATPase.     
Corre F, Jaxel C, Fuentes J, Menguy T, Falson P, Levine BA, Mller JV, Le Maire M
(2003) Ann N Y Acad Sci 986 : 90-5

121.  Regulation and mutational analysis of the HPr kinase/phosphorylase from Bacillus subtilis.     
Pompeo F, Granet Y, Lavergne JP, Grangeasse C, Nessler S, Jault JM, Galinier A
(2003) Biochemistry 42 : 6762-71

120.  The conserved glutamate residue adjacent to the Walker-B motif is the catalytic base for ATP hydrolysis in the ATP-binding cassette transporter BmrA.     
Orelle C, Dalmas O, Gros P, Di Pietro A, Jault JM
(2003) J Biol Chem 278 : 47002-8

119.  Overexpression of SERCA1a Ca2+-ATPase in yeast.     
Falson P, Lenoir G, Menguy T, Corre F, Montigny C, Pedersen PA, Thines D, Le Maire M
(2003) Ann N Y Acad Sci 986 : 312-4

118.  Modified jatrophane diterpenes as modulators of multidrug resistance from Euphorbia dendroides L.     
Corea G, Fattorusso E, Lanzotti V, Taglialatela-Scafati O, Appendino G, Ballero M, Simon PN, Dumontet C, Di Pietro A
(2003) Bioorg Med Chem 11 : 5221-7

117.  Purification of SERCA1a Ca2+-ATPase mutants expressed in yeast.     
Lenoir G, Montigny C, Le Maire M, Falson P
(2003) Ann N Y Acad Sci 986 : 333-4

116.  RU49953: a non-hormonal steroid derivative that potently inhibits P-glycoprotein and reverts cellular multidrug resistance.     
Perez-Victorias FJ, Conseil G, Munoz-Martinez F, Perez-Victoria JM, Dayan G, Marsaud V, Castanys S, Gamarro F, Renoir JM, Di Pietro A
(2003) Cell Mol Life Sci 60 : 526-35

115.  A new P-glycoprotein inhibitor from the caper spurge (Euphorbia lathyris).     
Appendino G, Della Porta C, Conseil G, Sterner O, Mercalli E, Dumontet C, Di Pietro A
(2003) J Nat Prod 66 : 140-2

2002 [Top] 11
114.  Interaction between the antiapoptotic protein Nr-13 and cytochrome c. Antagonistic effect of the BH3 domain of Bax.     
Moradi-Ameli M, Lorca T, Ficheux D, Di Pietro A, Gillet G
(2002) Biochemistry 41 : 8540-50

113.  4-Hydroxy-6-methoxyaurones with high-affinity binding to cytosolic domain of P-glycoprotein.     
Boumendjel A, Beney C, Deka N, Mariotte AM, Lawson MA, Trompier D, Baubichon-Cortay H, Di Pietro A
(2002) Chem Pharm Bull (Tokyo) 50 : 854-6

112.  Three-dimensional structure by cryo-electron microscopy of YvcC, an homodimeric ATP-binding cassette transporter from Bacillus subtilis.     
Chami M, Steinfels E, Orelle C, Jault JM, Di Pietro A, Rigaud JL, Marco S
(2002) J Mol Biol 315 : 1075-85

111.  Modulation by flavonoids of cell multidrug resistance mediated by P-glycoprotein and related ABC transporters.     
Di Pietro A, Conseil G, Perez-Victoria JM, Dayan G, Baubichon-Cortay H, Trompier D, Steinfels E, Jault JM, De Wet H, Maitrejean M, Comte G, Boumendjel A, Mariotte AM, Dumontet C, McIntosh DB, Goffeau A, Castanys S, Gamarro F, Barron D
(2002) Cell Mol Life Sci 59 : 307-22

110.  Multidrug resistance phenotype mediated by the P-glycoprotein-like transporter in Leishmania: a search for reversal agents.     
Perez-Victoria JM, Di Pietro A, Barron D, Ravelo AG, Castanys S, Gamarro F
(2002) Curr Drug Targets 3 : 311-33

109.  Overproduction in yeast and rapid and efficient purification of the rabbit SERCA1a Ca(2+)-ATPase.     
Lenoir G, Menguy T, Corre F, Montigny C, Pedersen PA, Thines D, Le Maire M, Falson P
(2002) Biochim Biophys Acta 1560 : 67-83

108.  Highly efficient over-production in E. coli of YvcC, a multidrug-like ATP-binding cassette transporter from Bacillus subtilis.     
Steinfels E, Orelle C, Dalmas O, Penin F, Miroux B, Di Pietro A, Jault JM
(2002) Biochim Biophys Acta 1565 : 1-5

107.  Insights into the functioning of Bacillus subtilis HPr kinase/phosphatase: affinity for its protein substrates and role of cations and phosphate.     
Lavergne JP, Jault JM, Galinier A
(2002) Biochemistry 41 : 6218-25

106.  A new family of phosphotransferases with a P-loop motif.     
Galinier A, Lavergne JP, Geourjon C, Fieulaine S, Nessler S, Jault JM
(2002) J Biol Chem 277 : 11362-7

105.  Recent advances in the discovery of flavonoids and analogs with high-affinity binding to P-glycoprotein responsible for cancer cell multidrug resistance.     
Boumendjel A, Di Pietro A, Dumontet C, Barron D
(2002) Med Res Rev 22 : 512-29

104.  Involvement of the cytoplasmic loop L6-7 in the entry mechanism for transport of Ca2+ through the sarcoplasmic reticulum Ca2+-ATPase.     
Menguy T, Corre F, Juul B, Bouneau L, Lafitte D, Derrick PJ, Sharma PS, Falson P, Levine BA, Mller JV, Le Maire M
(2002) J Biol Chem 277 : 13016-28

2001 [Top] 11
103.  Protein kinase C effectors bind to multidrug ABC transporters and inhibit their activity.     
Conseil G, Perez-Victoria JM, Jault JM, Gamarro F, Goffeau A, Hofmann J, Di Pietro A
(2001) Biochemistry 40 : 2564-71

102.  C-Isoprenylation of flavonoids enhances binding affinity toward P-glycoprotein and modulation of cancer cell chemoresistance.     
Comte G, Daskiewicz JB, Bayet C, Conseil G, Viornery-Vanier A, Dumontet C, Di Pietro A, Barron D
(2001) J Med Chem 44 : 763-8

101.  B-ring substituted 5,7-dihydroxyflavonols with high-affinity binding to P-glycoprotein responsible for cell multidrug resistance.     
Boumendjel A, Bois F, Beney C, Mariotte AM, Conseil G, Di Pietro A
(2001) Bioorg Med Chem Lett 11 : 75-7

100.  Sequence requirements of the ATP-binding site within the C-terminal nucleotide-binding domain of mouse P-glycoprotein: structure-activity relationships for flavonoid binding.     
De Wet H, McIntosh DB, Conseil G, Baubichon-Cortay H, Krell T, Jault JM, Daskiewicz JB, Barron D, Di Pietro A
(2001) Biochemistry 40 : 10382-91

99.  High-affinity binding of silybin derivatives to the nucleotide-binding domain of a Leishmania tropica P-glycoprotein-like transporter and chemosensitization of a multidrug-resistant parasite to daunomycin.     
Perez-Victoria JM, Perez-Victoria FJ, Conseil G, Maitrejean M, Comte G, Barron D, Di Pietro A, Castanys S, Gamarro F
(2001) Antimicrob Agents Chemother 45 : 439-46

98.  Modulation of cancer cell multidrug resistance by an extract of Ficus citrifolia.     
Simon PN, Chaboud A, Darbour N, Di Pietro A, Dumontet C, Lurel F, Raynaud J, Barron D
(2001) Anticancer Res 21 : 1023-7

97.  MDR1 causes resistance to the antitumour drug miltefosine.   
Rybczynska M, Liu R, Lu P, Sharom FJ, Steinfels E, Pietro AD, Spitaler M, Grunicke H, Hofmann J
(2001) Br J Cancer 84 : 1405-11

96.  SERCA1 truncated proteins unable to pump calcium reduce the endoplasmic reticulum calcium concentration and induce apoptosis.     
Chami M, Gozuacik D, Lagorce D, Brini M, Falson P, Peaucellier G, Pinton P, Lecoeur H, Gougeon ML, Le Maire M, Rizzuto R, Brechot C, Paterlini-Brechot P
(2001) J Cell Biol 153 : 1301-14

95.  A common mechanism for ATP hydrolysis in ABC transporter and helicase superfamilies.     
Geourjon C, Orelle C, Steinfels E, Blanchet C, Deleage G, Di Pietro A, Jault JM
(2001) Trends Biochem Sci 26 : 539-44

94.  Natural and synthetic benzophenones: interaction with the cytosolic binding domain of P-glycoprotein.     
Rancon S, Chaboud A, Darbour N, Comte G, Bayet C, Simon PN, Raynaud J, Di Pietro A, Cabalion P, Barron D
(2001) Phytochemistry 57 : 553-7

93.  The "catalytic" triad of isocitrate dehydrogenase kinase/phosphatase from E. coli and its relationship with that found in eukaryotic protein kinases.     
Oudot C, Cortay JC, Blanchet C, Laporte DC, Di Pietro A, Cozzone AJ, Jault JM
(2001) Biochemistry 40 : 3047-55

2000 [Top] 7
92.  The flavanolignan silybin and its hemisynthetic derivatives, a novel series of potential modulators of P-glycoprotein.     
Maitrejean M, Comte G, Barron D, El Kirat K, Conseil G, Di Pietro A
(2000) Bioorg Med Chem Lett 10 : 157-60

91.  Evidence for a second nucleotide binding site in rat elongation factor eEF-2 specific for adenylic nucleotides.     
Gonzalo P, Sontag B, Lavergne JP, Jault JM, Reboud JP
(2000) Biochemistry 39 : 13558-64

90.  Hepatitis B virus-related insertional mutagenesis implicates SERCA1 gene in the control of apoptosis.     
Chami M, Gozuacik D, Saigo K, Capiod T, Falson P, Lecoeur H, Urashima T, Beckmann J, Gougeon ML, Claret M, Le Maire M, Brechot C, Paterlini-Brechot P
(2000) Oncogene 19 : 2877-86

89.  Prenylated xanthones as potential P-glycoprotein modulators.     
Tchamo DN, Dijoux-Franca MG, Mariotte AM, Tsamo E, Daskiewicz JB, Bayet C, Barron D, Conseil G, Di Pietro A
(2000) Bioorg Med Chem Lett 10 : 1343-5

88.  The HPr kinase from Bacillus subtilis is a homo-oligomeric enzyme which exhibits strong positive cooperativity for nucleotide and fructose 1,6-bisphosphate binding.     
Jault JM, Fieulaine S, Nessler S, Gonzalo P, Di Pietro A, Deutscher J, Galinier A
(2000) J Biol Chem 275 : 1773-80

87.  Clean Western blots of membrane proteins after yeast heterologous expression following a shortened version of the method of Perini et al.     
Fuentes JM, Lompre AM, Mller JV, Falson P, Le Maire M
(2000) Anal Biochem 285 : 276-8

86.  Prenyl-flavonoids as potent inhibitors of the Pdr5p multidrug ABC transporter from Saccharomyces cerevisiae.     
Conseil G, Decottignies A, Jault JM, Comte G, Barron D, Goffeau A, Di Pietro A
(2000) Biochemistry 39 : 6910-7

1999 [Top] 4
85.  Heterologous expression of the red-cell anion exchanger (band 3; AE1).     
Groves JD, Parker MD, Askin D, Falson P, Le Maire M, Tanner MJ
(1999) Biochem Soc Trans 27 : 917-23

84.  The isocitrate dehydrogenase kinase/phosphatase from Escherichia coli is highly sensitive to in-vitro oxidative conditions role of cysteine67 and cysteine108 in the formation of a disulfide-bonded homodimer.     
Oudot C, Jaquinod M, Cortay JC, Cozzone AJ, Jault JM
(1999) Eur J Biochem 262 : 224-9

83.  P-glycoprotein-mediated resistance to chemotherapy in cancer cells: using recombinant cytosolic domains to establish structure-function relationships.     
Di Pietro A, Dayan G, Conseil G, Steinfels E, Krell T, Trompier D, Baubichon-Cortay H, Jault J
(1999) Braz J Med Biol Res 32 : 925-39

82.  Correlation between the affinity of flavonoids binding to the cytosolic site of Leishmania tropica multidrug transporter and their efficiency to revert parasite resistance to daunomycin.     
Perez-Victoria JM, Chiquero MJ, Conseil G, Dayan G, Di Pietro A, Barron D, Castanys S, Gamarro F
(1999) Biochemistry 38 : 1736-43

1998 [Top] 7
81.  Mutagenesis of the fructose-6-phosphate-binding site in the 2-kinase domain of 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase.     
Bertrand L, Vertommen D, Freeman PM, Wouters J, Depiereux E, Di Pietro A, Hue L, Rider MH
(1998) Eur J Biochem 254 : 490-6

80.  Halogenated chalcones with high-affinity binding to P-glycoprotein: potential modulators of multidrug resistance.     
Bois F, Beney C, Boumendjel A, Mariotte AM, Conseil G, Di Pietro A
(1998) J Med Chem 41 : 4161-4

79.  The cytoplasmic loop located between transmembrane segments 6 and 7 controls activation by Ca2+ of sarcoplasmic reticulum Ca2+-ATPase.     
Menguy T, Corre F, Bouneau L, Deschamps S, Mller JV, Champeil P, Le Maire M, Falson P
(1998) J Biol Chem 273 : 20134-43

78.  Inactivation of isocitrate dehydrogenase kinase/phosphatase by 5'-[p-(fluorosulfonyl)benzoyl]adenosine is not due to the labeling of the invariant lysine residue found in the protein kinase family.     
Oudot C, Jault JM, Jaquinod M, Negre D, Prost JF, Cozzone AJ, Cortay JC
(1998) Eur J Biochem 258 : 579-85

77.  Ligand binding to macromolecules or micelles: use of centrifugal ultrafiltration to measure low-affinity binding.     
Menguy T, Chenevois S, Guillain F, Le Maire M, Falson P, Champeil P
(1998) Anal Biochem 264 : 141-8

76.  Flavonoids: a class of modulators with bifunctional interactions at vicinal ATP- and steroid-binding sites on mouse P-glycoprotein.     
Conseil G, Baubichon-Cortay H, Dayan G, Jault JM, Barron D, Di Pietro A
(1998) Proc Natl Acad Sci U S A 95 : 9831-6

75.  Characterization of a protease-resistant domain of the cytosolic portion of sarcoplasmic reticulum Ca2+-ATPase. Nucleotide- and metal-binding sites.     
Champeil P, Menguy T, Soulie S, Juul B, De Gracia AG, Rusconi F, Falson P, Denoroy L, Henao F, Le Maire M, Moller JV
(1998) J Biol Chem 273 : 6619-31

1997 [Top] 7
74.  Site-directed mutagenesis of Lys-174, Asp-179 and Asp-191 in the 2-kinase domain of 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase.     
Bertrand L, Deprez J, Vertommen D, Di Pietro A, Hue L, Rider MH
(1997) Biochem J 321 ( Pt 3) : 623-7

73.  Probing of the membrane topology of sarcoplasmic reticulum Ca2+-ATPase with sequence-specific antibodies. Evidence for plasticity of the c-terminal domain.     
Moller JV, Ning G, Maunsbach AB, Fujimoto K, Asai K, Juul B, Lee YJ, Gomez De Gracia A, Falson P, Le Maire M
(1997) J Biol Chem 272 : 29015-32

72.  The cytoplasmic loop between putative transmembrane segments 6 and 7 in sarcoplasmic reticulum Ca2+-ATPase binds Ca2+ and is functionally important.     
Falson P, Menguy T, Corre F, Bouneau L, De Gracia AG, Soulie S, Centeno F, Moller JV, Champeil P, Le Maire M
(1997) J Biol Chem 272 : 17258-62

71.  Binding of steroid modulators to recombinant cytosolic domain from mouse P-glycoprotein in close proximity to the ATP site.     
Dayan G, Jault JM, Baubichon-Cortay H, Baggetto LG, Renoir JM, Baulieu EE, Gros P, Di Pietro A
(1997) Biochemistry 36 : 15208-15

70.  Complete removal and exchange of sodium dodecyl sulfate bound to soluble and membrane proteins and restoration of their activities, using ceramic hydroxyapatite chromatography.     
Dong M, Baggetto LG, Falson P, Le Maire M, Penin F
(1997) Anal Biochem 247 : 333-41

69.  Probing of membrane topology and stability of sarcoplasmic reticulum Ca(2+)-ATPase and Na+,K+ -ATPase with sequence-specific antibodies.     
Mller JV, Juul B, Falson P, Le Maire M
(1997) Ann N Y Acad Sci 834 : 142-5

68.  Mutagenesis of charged residues in a conserved sequence in the 2-kinase domain of 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase.     
Bertrand L, Vertommen D, Feytmans E, Di Pietro A, Rider MH, Hue L
(1997) Biochem J 321 ( Pt 3) : 609-14

1996 [Top] 6
67.  Recombinant N-terminal nucleotide-binding domain from mouse P-glycoprotein. Overexpression, purification, and role of cysteine 430.     
Dayan G, Baubichon-Cortay H, Jault JM, Cortay JC, Deleage G, Di Pietro A
(1996) J Biol Chem 271 : 11652-8

66.  Does the gamma subunit move to an abortive position for ATP hydrolysis when the F-1 center dot ADP center dot Mg complex isomerizes to the inactive F-1*center dot ADP center dot Mg complex?   
Allison WS, Jault JM, Dou C, Grodsky NB
(1996) J Bioenerg Biomembr 28 : 433-438

65.  Functional cell surface expression of the anion transport domain of human red cell band 3 (AE1) in the yeast Saccharomyces cerevisiae.     
Groves JD, Falson P, Le Maire M, Tanner MJ
(1996) Proc Natl Acad Sci U S A 93 : 12245-50

64.  Urea reduces the aggregation of membrane proteins on sodium dodecyl sulfate-polyacrylamide gel electrophoresis.     
Soulie S, Mller JV, Falson P, Le Maire M
(1996) Anal Biochem 236 : 363-4

63.  The ATP-binding site in the 2-kinase domain of liver 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase. Study of the role of Lys-54 and Thr-55 by site-directed mutagenesis.     
Vertommen D, Bertrand L, Sontag B, Di Pietro A, Louckx MP, Vidal H, Hue L, Rider MH
(1996) J Biol Chem 271 : 17875-80

62.  The alpha(3)beta(3)gamma subcomplex of the F-1-ATPase from the thermophilic Bacillus PS3 with the beta T165S substitution does not entrap inhibitory MgADP in a catalytic site during turnover   
Jault JM, Dou C, Grodsky NB,Matsui T, Yoshida M, Allison WS
(1996) J Biol Chem 271 :  28818-28824

1995 [Top] 2
61.  CYTOMEGALOVIRUS-INFECTION INDUCES HIGH-LEVELS OF CYCLINS, PHOSPHORYLATED RB, AND P53, LEADING TO CELL-CYCLE ARREST   
JAULT FM, JAULT JM, RUCHTI F, FORTUNATO EA, CLARK C, CORBEIL J, RICHMAN DD, SPECTOR DH
(1995) J Virol 69 : 6697-6704

60.  The alpha(3)beta(3)gamma complex of the F-1-ATPase from thermophilic Bacillus PS3 containing the alpha D261N substitution fails to dissociate inhibitory MgADP from a catalytic site when ATP binds to noncatalytic sites   
Jault JM, Matsui T, Jault FM, Kaibara C, Muneyuki E, Yoshida M, Kagawa Y, Allison WS
(1995) Biochemistry 34 : 16412-16418

1994 [Top] 9
59.  ADP TETHERED TO TYROSINE-BETA-345 AT THE CATALYTIC SITE OF THE BOVINE HEART F1-ATPASE IS CONVERTED TO TETHERED AMP BY MG2+-DEPENDENT HYDROLYSIS WHEN THE ENZYME IS PHOTOINACTIVATED WITH 2-N-3-ADP   
JAULT JM, ALLISON WS
(1994) FEBS Lett 347 : 13-16

58.  Expression of the sarcoplasmic reticulum Ca(2+)-ATPase in yeast.     
Centeno F, Deschamps S, Lompre AM, Anger M, Moutin MJ, Dupont Y, Palmgren MG, Villalba JM, Mller JV, Falson P
(1994) FEBS Lett 354 : 117-22

57.  Preparation of highly phosphorylating mitochondria from the yeast Schizosaccharomyces pombe.     
Jault JM, Comte J, Gautheron DC, Di Pietro A
(1994) J Bioenerg Biomembr 26 : 447-56

56.  PROBING THE SPECIFICITY OF NUCLEOTIDE-BINDING TO THE F1-ATPASE FROM THERMOPHILIC BACILLUS PS3 AND ITS ISOLATED ALPHA-SUBUNIT AND BETA-SUBUNIT WITH 2-N3-[BETA,GAMMA-P-32]ATP   
JAULT JM, KAIBARA C, YOSHIDA M, GARROD S, ALLISON WS
(1994) Arch Biochem Biophys 310 : 282-288

55.  INHIBITION AND INACTIVATION OF THE F(1)-ADENOSINE-TRIPHOSPHATASE FROM BACILLUS PS3 BY DEQUALINIUM AND ACTIVATION OF THE ENZYME BY LAURYL DIMETHYLAMINE OXIDE   
PAIK SR, JAULT JM, ALLISON WS
(1994) BIOCHEMISTRY 33 : 126-133

54.  Overexpression and purification of the carboxyl-terminal nucleotide-binding domain from mouse P-glycoprotein. Strategic location of a tryptophan residue.     
Baubichon-Cortay H, Baggetto LG, Dayan G, Di Pietro A
(1994) J Biol Chem 269 : 22983-9

53.  HYSTERETIC INHIBITION OF THE BOVINE HEART MITOCHONDRIAL F1-ATPASE IS DUE TO SATURATION OF NONCATALYTIC SITES WITH ADP WHICH BLOCKS ACTIVATION OF THE ENZYME BY ATP   
JAULT JM, ALLISON WS
(1994) J Biol Chem 269 : 319-325

52.  CATALYTIC COOPERATIVITY OF BEEF-HEART MITOCHONDRIAL F1-ATPASE REVEALED BY USING 2',3'-O-(2,4,6-TRINITROPHENYL)-ATP AS A SUBSTRATE - AN INDICATION OF MUTUALLY ACTIVATING CATALYTIC SITES   
MUNEYUKI E, HISABORI T, ALLISON WS, JAULT JM, SASAYAMA T, YOSHIDA M
(1994) BIOCHIMICA ET BIOPHYSICA ACTA-BIOENERGETICS 1188 : 108-116

51.  LOWERED TEMPERATURE OR BINDING OF PYROPHOSPHATE TO SITES FOR NONCATALYTIC NUCLEOTIDES MODULATES THE ATPASE ACTIVITY OF THE BEEF-HEART MITOCHONDRIAL F1-ATPASE BY DECREASING THE AFFINITY OF A CATALYTIC SITE FOR INHIBITORY MGADP   
JAULT JM, PAIK SR, GRODSKY NB, ALLISON WS
(1994) BIOCHEMISTRY 33 : 14979-14985

1993 [Top] 7
50.  Chemical modification of alpha-subunit tryptophan residues in Schizosaccharomyces pombe mitochondrial F1 adenosine 5'-triphosphatase: differential reactivity and role in activity.     
Divita G, Jault JM, Gautheron DC, Di Pietro A
(1993) Biochemistry 32 : 1017-24

49.  Glutamine 170 to tyrosine substitution in yeast mitochondrial F1 beta-subunit increases catalytic site interaction with GDP and IDP and produces negative cooperativity of GTP and ITP hydrolysis.     
Jault JM, Divita G, Allison WS, Di Pietro A
(1993) J Biol Chem 268 : 20762-7

48.  Intrinsic tryptophan fluorescence of rat liver elongation factor eEF-2 to monitor the interaction with guanylic and adenylic nucleotides and related conformational changes.     
Sontag B, Reboud AM, Divita G, Di Pietro A, Guillot D, Reboud JP
(1993) Biochemistry 32 : 1976-80

47.  Structural mapping of catalytic site with respect to alpha-subunit and noncatalytic site in yeast mitochondrial F1-ATPase using fluorescence resonance energy transfer.     
Divita G, Goody RS, Gautheron DC, Di Pietro A
(1993) J Biol Chem 268 : 13178-86

46.  SLOW BINDING OF ATP TO NONCATALYTIC NUCLEOTIDE BINDING-SITES WHICH ACCELERATES CATALYSIS IS RESPONSIBLE FOR APPARENT NEGATIVE COOPERATIVITY EXHIBITED BY THE BOVINE MITOCHONDRIAL F1-ATPASE   
JAULT JM, ALLISON WS
(1993) J Biol Chem 268 : 1558-1566

45.  Functional nucleotide-binding domain in the F0F1-ATPsynthase alpha subunit from the yeast Schizosaccharomyces pombe.     
Falson P, Penin F, Divita G, Lavergne JP, Di Pietro A, Goody RS, Gautheron DC
(1993) Biochemistry 32 : 10387-97

44.  GTP binding to elongation factor eEF-2 unmasks a tryptophan residue required for biological activity.     
Guillot D, Penin F, Di Pietro A, Sontag B, Lavergne JP, Reboud JP
(1993) J Biol Chem 268 : 20911-6

1992 [Top] 4
43.  An efficient procedure to dialyze volumes in the range of 10-200 microliters.     
Falson P
(1992) Biotechniques 13 : 20-2

42.  Histone H1a subtype presents structural differences compared to other histone H1 subtypes. Evidence for a specific motif in the C-terminal domain.     
Baubichon-Cortay H, Mallet L, Denoroy L, Roux B
(1992) Biochim Biophys Acta 1122 : 167-77

41.  FUNCTIONAL SITES IN F1-ATPASES - LOCATION AND INTERACTIONS   
ALLISON WS, JAULT JM, ZHUO SQ, PAIK SR
(1992) J Bioenerg Biomembr 24 : 469-477

40.  Differential nucleotide binding to catalytic and noncatalytic sites and related conformational changes involving alpha/beta-subunit interactions as monitored by sensitive intrinsic fluorescence in Schizosaccharomyces pombe mitochondrial F1.     
Divita G, Di Pietro A, Roux B, Gautheron DC
(1992) Biochemistry 31 : 5791-8

1991 [Top] 6
39.  Beta subunit of mitochondrial F1-ATPase from the fission yeast. Deduced sequence of the wild type protein and identification of a mutation that increases nucleotide binding.     
Falson P, Leterme S, Capiau C, Boutry M
(1991) Eur J Biochem 200 : 61-7

38.  Alteration of apparent negative cooperativity of ATPase activity by alpha-subunit glutamine 173 mutation in yeast mitochondrial F1. Correlation with impaired nucleotide interaction at a regulatory site.     
Jault JM, Di Pietro A, Falson P, Gautheron DC
(1991) J Biol Chem 266 : 8073-8

37.  Intrinsic tryptophan fluorescence of Schizosaccharomyces pombe mitochondrial F1-ATPase. A powerful probe for phosphate and nucleotide interactions.     
Divita G, Di Pietro A, Deleage G, Roux B, Gautheron DC
(1991) Biochemistry 30 : 3256-62

36.  Alpha subunit of mitochondrial F1-ATPase from the fission yeast. Deduced sequence of the wild type and identification of a mutation that alters apparent negative cooperativity.     
Falson P, Maffey L, Conrath K, Boutry M
(1991) J Biol Chem 266 : 287-93

35.  Sialylation processes in mitochondria: evidence for two distinct sialyltransferases located in the outer membrane.     
Gasnier F, Baubichon-Cortay H, Louisot P, Gateau-Roesch O
(1991) J Biochem 110 : 702-7

34.  Glycoprotein sialyltransferases in eucaryotic cells.     
Broquet P, Baubichon-Cortay H, George P, Louisot P
(1991) Int J Biochem 23 : 385-9

1990 [Top] 1
33.  Effect of desipramine on a glycoprotein sialyltransferase activity in C6 cultured glioma cells.     
Broquet P, Baubichon-Cortay H, George P, Peschard MJ, Louisot P
(1990) J Neurochem 54 : 388-94

1989 [Top] 5
32.  Different reactivity of two brain sialyltransferases towards sulfhydryl reagents. Evidence for a thiol group involved in the nucleotide-sugar binding site of the NeuAc alpha 2-3Gal beta 1-3GalNAc alpha(2-6)sialyltransferase.     
Baubichon-Cortay H, Broquet P, George P, Louisot P
(1989) Glycoconj J 6 : 115-27

31.  Purification from a yeast mutant of mitochondrial F1 with modified beta-subunit. High affinity for nucleotides and high negative cooperativity of ATPase activity.     
Falson P, Di Pietro A, Jault JM, Gautheron DC, Boutry M
(1989) Biochim Biophys Acta 975 : 119-26

30.  Evidence for an O-glycan sialylation system in brain. Characterization of a beta-galactoside alpha 2,3-sialyltransferase from rat brain regulating the expression of an alpha-N-acetylgalactosaminide alpha 2,6-sialyltransferase activity.     
Baubichon-Cortay H, Broquet P, George P, Louisot P
(1989) Eur J Biochem 182 : 257-65

29.  Structure-function relationships of mitochondrial ATPase-ATPsynthase using Schizosaccharomyces pombe yeast mutants with altered F1 subunits.     
Di Pietro A, Jault JM, Falson P, Divita G, Gautheron DC
(1989) Biochimie 71 : 931-40

28.  A yeast strain with mutated beta-subunits of mitochondrial ATPase-ATPsynthase: high azide and bicarbonate sensitivity of the ATPase activity.     
Jault JM, Di Pietro A, Falson P, Gautheron DC, Boutry M, Goffeau A
(1989) Biochem Biophys Res Commun 158 : 392-9

1988 [Top] 2
27.  Fate of nucleotides bound to reconstituted Fo-F1 during adenosine 5'-triphosphate synthesis activation or hydrolysis: role of protein inhibitor and hysteretic inhibition.     
Penin F, Di Pietro A, Godinot C, Gautheron DC
(1988) Biochemistry 27 : 8969-74

26.  IF1 inhibition of mitochondrial F1-ATPase is correlated to entrapment of four adenine- or guanine-nucleotides including at least one triphosphate.     
Di Pietro A, Penin F, Julliard JH, Godinot C, Gautheron DC
(1988) Biochem Biophys Res Commun 152 : 1319-25

1987 [Top] 2
25.  Revertant of the yeast Schizosaccharomyces pombe with modified alpha subunits of mitochondrial ATPase-ATPsynthase: impaired nucleotide interactions with soluble and membrane-bound enzyme.     
Falson P, Di Pietro A, Darbouret D, Jault JM, Gautheron DC, Boutry M, Goffeau A
(1987) Biochem Biophys Res Commun 148 : 1182-8

24.  Study of circadian correlations between acetylcholine muscarinic receptor and brain glycosyltransferases by multivariate analysis.     
Broquet P, Martin A, Peschard MJ, Baubichon-Cortay H, Serres-Guillaumond M, Louisot P
(1987) Int J Biochem 19 : 653-6

1986 [Top] 6
23.  A brain sialyltransferase having a narrow specificity for O-glycosyl-linked oligosaccharide chains.     
Baubichon-Cortay H, Serres-Guillaumond M, Louisot P, Broquet P
(1986) Carbohydr Res 149 : 209-23

22.  Role of phosphate on the ADP-induced hysteretic inhibition of mitochondrial adenosine 5'-triphosphatase. Effects of the natural protein inhibitor.     
Di Pietro A, Fellous G, Godinot C, Gautheron DC
(1986) Biochim Biophys Acta 851 : 283-94

21.  Different reactivity to lysophosphatidylcholine, DIDS and trypsin of two brain sialyltransferases specific for O-glycans: a consequence of their topography in the endoplasmic membranes.     
Baubichon-Cortay H, Serres-Guillaumond M, Broquet P, Louisot P
(1986) Biochim Biophys Acta 862 : 243-53

20.  Structure and function of the ATPase-ATP synthase complex of mitochondria as compared to chloroplasts and bacteria.     
Godinot C, Di Pietro A
(1986) Biochimie 68 : 367-74

19.  Chemical modification of thiol groups of mitochondrial F1-ATPase from the yeast Schizosaccharomyces pombe. Involvement of alpha- and gamma-subunits in the enzyme activity.     
Falson P, Di Pietro A, Gautheron DC
(1986) J Biol Chem 261 : 7151-9

18.  Chemical modification of essential carboxyl group and histidine residue in the plasma-membrane 5'-nucleotidase.     
Harb J, Meflah K, Di Pietro A, Bernard S, Gautheron DC
(1986) Biochim Biophys Acta 870 : 320-6

1985 [Top] 2
17.  Essential arginyl residues in the H+-translocating ATPase of plasma membrane from the yeast Schizosaccharomyces pombe.     
Di Pietro A, Goffeau A
(1985) Eur J Biochem 148 : 35-9

16.  The RNA polymerase I initiation site and the external transcribed spacer of the fission yeast Schizosaccharomyces pombe ribosomal RNA genes.     
Balzi E, Di Pietro A, Goffeau A, Van Heerikhuizen H, Klootwijk J
(1985) Gene 39 : 165-72

1984 [Top] 1
15.  Subcellular localisation of cerebral fucosyltransferase.     
Broquet P, Serres-Guillaumond M, Baubichon-Cortay H, Peschard MJ, Louisot P
(1984) FEBS Lett 174 : 43-6

1983 [Top] 1
14.  Use of trypsin to monitor conformational changes of mitochondrial adenosinetriphosphatase induced by nucleotides and phosphate.     
Di Pietro A, Godinot C, Gautheron DC
(1983) Biochemistry 22 : 785-92

1982 [Top] 1
13.  Abolition of anion-activation of mitochondrial F1-ATPase by the partial ADP-induced hysteretic inhibition.     
Baubichon H, Di Pietro A, Godinot C, Gautheron DC
(1982) FEBS Lett 137 : 261-4

1981 [Top] 2
12.  Interaction between catalytic and regulatory sites of mitochondrial F1 adenosine-5'-triphosphatase as monitored by the differential effects of inhibitors and nucleotide analogues on the "hysteretic" behavior of the enzyme.     
Di Pietro A, Godinot C, Gautheron DC
(1981) Biochemistry 20 : 6312-8

11.  Competition between ADP and nucleotide analogues to occupy regulatory sites(s) related to hysteretic inhibition of mitochondrial F1-ATPase.     
Baubichon H, Godinot C, Di Pietro A, Gautheron DC
(1981) Biochem Biophys Res Commun 100 : 1032-8

1980 [Top] 2
10.  "Hysteric" behavior and nucleotide binding sites of pig heart mitochondrial F1 adenosine 5'-triphosphatase.     
Di Pietro A, Penin F, Godinot C, Gautheron DC
(1980) Biochemistry 19 : 5671-8

9.  Role of magnesium on kinetic parameters of soluble F1-ATPase from pig heart mitochondria.     
Fleury B, Di Pietro A, Godinot C, Gautheron DC
(1980) Biochimie 62 : 733-7

1979 [Top] 1
8.  Affinity labeling of catalytic and regulatory sites of pig heart mitochondrial F1-ATPase by 5'-p-fluorosulfonylbenzoyladenosine.     
Di Pietro A, Godinot C, Martin JC, Gautheron DC
(1979) Biochemistry 18 : 1738-45

1978 [Top] 1
7.  [Kinetic study of membrane 5'-nucleotidase activity in cultured diploid cells].   
Daveze JL, Di Pietro A, Frappa J, Deloince R, Beaudry Y, Fontanges R
(1978) C R Acad Sci Hebd Seances Acad Sci D 286 : 1621-4

1977 [Top] 4
6.  Binding of the polyflavane P13 on various pig myocardial membranes--effects on protein release and on Ca2+ and Mg2+ movements.     
Di Pietro A, Godinot C, Vial C, Gautheron DC
(1977) Biochem Pharmacol 26 : 1775-81

5.  [Early effect of poliomyelitis virus on 5'-nucleotidase activity in HeLa cells].   
Di Pietro A, Deloince R, Beaudry Y, Fontanges R
(1977) C R Acad Sci Hebd Seances Acad Sci D 285 : 925-8

4.  Effects of P13, a polyflavane compound, on pig myocardium ATP-synthesis, ATPases and creatine kinase.     
Di Pietro A, Godinot C, Gautheron DC, Foulhoux P
(1977) Biochem Pharmacol 26 : 1021-6

3.  Vicinal dithiol in pig heart mitochondrial F1-ATPase related to thermal or ATP-dependent conformational changes.     
Godinot C, Di Pietro A, Blanchy B, Penin F, Gautheron DC
(1977) J Bioenerg Biomembr 9 : 255-69

1975 [Top] 2
2.  Masking of co-operativity of nucleotide sites in pig heart mitochondrial ATPase (F1) by heating.     
Godinot C, Di Pietro A, Gautheron DC
(1975) FEBS Lett 60 : 250-5

1.  Pig heart mitochondrial ATPase : properties of purified and membrane-bound enzyme. Effects of flavonoids.     
Di Pietro A, Godinot C, Bouillant ML, Gautheron DC
(1975) Biochimie 57 : 959-67